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Fate of nanostructured lipid carriers (NLCs) following the oral route: design, pharmacokinetics and biodistribution

Bibliographic reference Beloqui Garcia, Ana ; Solinís, María Ángeles ; Delgado, Araceli ; Evora, Carmen ; Isla, Arantxazu ; et. al. Fate of nanostructured lipid carriers (NLCs) following the oral route: design, pharmacokinetics and biodistribution. In: Journal of Microencapsulation, Vol. 31, no. 1, p. 1-8 (2014)
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  1. ABDELWAHED W, DEGOBERT G, STAINMESSE S, FESSI H, Freeze-drying of nanoparticles: Formulation, process and storage considerations☆, 10.1016/j.addr.2006.09.017
  2. N’Goma Jean-Claude Bakala, Amara Sawsan, Dridi Kaouthar, Jannin Vincent, Carrière Frédéric, Understanding the lipid-digestion processes in the GI tract before designing lipid-based drug-delivery systems, 10.4155/tde.11.138
  3. Chakraborty Subhashis, Shukla Dali, Mishra Brahmeshwar, Singh Sanjay, Lipid – An emerging platform for oral delivery of drugs with poor bioavailability, 10.1016/j.ejpb.2009.06.001
  4. Charman WN, Lymphatic transport of drugs (1992)
  5. Chen Mei-Ling, Lipid excipients and delivery systems for pharmaceutical development: A regulatory perspective, 10.1016/j.addr.2007.09.010
  6. Chen Chih-Chieh, Tsai Tung-Hu, Huang Zih-Rou, Fang Jia-You, Effects of lipophilic emulsifiers on the oral administration of lovastatin from nanostructured lipid carriers: Physicochemical characterization and pharmacokinetics, 10.1016/j.ejpb.2009.12.008
  7. Dahan Arik, Hoffman Amnon, The effect of different lipid based formulations on the oral absorption of lipophilic drugs: The ability of in vitro lipolysis and consecutive ex vivo intestinal permeability data to predict in vivo bioavailability in rats, 10.1016/j.ejpb.2007.01.017
  8. Dahan Arik, Hoffman Amnon, Rationalizing the selection of oral lipid based drug delivery systems by an in vitro dynamic lipolysis model for improved oral bioavailability of poorly water soluble drugs, 10.1016/j.jconrel.2008.03.021
  9. Das Surajit, Chaudhury Anumita, Recent Advances in Lipid Nanoparticle Formulations with Solid Matrix for Oral Drug Delivery, 10.1208/s12249-010-9563-0
  10. del Pozo-Rodríguez A., Solinís M.A., Gascón A.R., Pedraz J.L., Short- and long-term stability study of lyophilized solid lipid nanoparticles for gene therapy, 10.1016/j.ejpb.2008.09.015
  11. Florence Alexander T., Nanoparticle uptake by the oral route: Fulfilling its potential?, 10.1016/j.ddtec.2005.05.019
  12. Florence Alexander T, Hussain Nasir, Transcytosis of nanoparticle and dendrimer delivery systems: evolving vistas, 10.1016/s0169-409x(01)00184-3
  13. Hauss David J., Oral lipid-based formulations, 10.1016/j.addr.2007.05.006
  14. Jannin V., Musakhanian J., Marchaud D., Approaches for the development of solid and semi-solid lipid-based formulations, 10.1016/j.addr.2007.09.006
  15. Kesisoglou Filippos, Panmai Santipharp, Wu Yunhui, Nanosizing — Oral formulation development and biopharmaceutical evaluation, 10.1016/j.addr.2007.05.003
  16. Konan Yvette N, Gurny Robert, Allémann Eric, Preparation and characterization of sterile and freeze-dried sub-200 nm nanoparticles, 10.1016/s0378-5173(01)00944-9
  17. Krishnaiah YSR, J Bioequiv Availab, 2, 28 (2010)
  18. Langguth P., Hanafy A., Frenzel D., Grenier P., Nhamias A., Ohlig T., Vergnault G., Spahn-Langguth H., Nanosuspension Formulations for Low-Soluble Drugs: Pharmacokinetic Evaluation Using Spironolactone as Model Compound, 10.1081/ddc-52182
  19. Limayem Blouza I., Charcosset C., Sfar S., Fessi H., Preparation and characterization of spironolactone-loaded nanocapsules for paediatric use, 10.1016/j.ijpharm.2006.06.022
  20. Mehnert W, Solid lipid nanoparticles Production, characterization and applications, 10.1016/s0169-409x(01)00105-3
  21. Merisko-Liversidge Elaine M., Liversidge Gary G., Drug Nanoparticles: Formulating Poorly Water-Soluble Compounds, 10.1177/0192623307310946
  22. Merisko-Liversidge Elaine, Liversidge Gary G., Nanosizing for oral and parenteral drug delivery: A perspective on formulating poorly-water soluble compounds using wet media milling technology, 10.1016/j.addr.2010.12.007
  23. Merisko-Liversidge Elaine, Liversidge Gary G, Cooper Eugene R, Nanosizing: a formulation approach for poorly-water-soluble compounds, 10.1016/s0928-0987(02)00251-8
  24. Muchow Marc, Maincent Philippe, Müller Rainer H., Lipid Nanoparticles with a Solid Matrix (SLN®, NLC®, LDC®) for Oral Drug Delivery, 10.1080/03639040802130061
  25. Müller R, Solid lipid nanoparticles (SLN) for controlled drug delivery – a review of the state of the art, 10.1016/s0939-6411(00)00087-4
  26. Müller R.H, Radtke M, Wissing S.A, Nanostructured lipid matrices for improved microencapsulation of drugs, 10.1016/s0378-5173(02)00180-1
  27. Müller R.H., Runge S., Ravelli V., Mehnert W., Thünemann A.F., Souto E.B., Oral bioavailability of cyclosporine: Solid lipid nanoparticles (SLN®) versus drug nanocrystals, 10.1016/j.ijpharm.2006.02.045
  28. Müllertz Anette, Ogbonna Anayo, Ren Shan, Rades Thomas, New perspectives on lipid and surfactant based drug delivery systems for oral delivery of poorly soluble drugs : Lipid and surfactant drug delivery systems, 10.1111/j.2042-7158.2010.01107.x
  29. O'Driscoll C.M., Griffin B.T., Biopharmaceutical challenges associated with drugs with low aqueous solubility—The potential impact of lipid-based formulations, 10.1016/j.addr.2007.10.012
  30. Overdiek H.W.P.M., Merkus F.W.H.M., THE METABOLISM AND BIOPHARMACEUTICS OF SPIRONOLACTONE IN MAN, 10.1515/dmdi.1987.5.4.273
  31. Porter Christopher J. H., Trevaskis Natalie L., Charman William N., Lipids and lipid-based formulations: optimizing the oral delivery of lipophilic drugs, 10.1038/nrd2197
  32. Porter Christopher J.H., Pouton Colin W., Cuine Jean F., Charman William N., Enhancing intestinal drug solubilisation using lipid-based delivery systems, 10.1016/j.addr.2007.10.014
  33. Pouton Colin W., Formulation of poorly water-soluble drugs for oral administration: Physicochemical and physiological issues and the lipid formulation classification system, 10.1016/j.ejps.2006.04.016
  34. Pouton Colin W., Porter Christopher J.H., Formulation of lipid-based delivery systems for oral administration: Materials, methods and strategies, 10.1016/j.addr.2007.10.010
  35. Saha Gopal B., Fundamentals of Nuclear Pharmacy, ISBN:9781441958594, 10.1007/978-1-4419-5860-0
  36. Szymendera J, J Nucl Med, 15, 314 (1974)
  37. Tarr Bryan D., Yalkowsky Samuel H., 10.1023/a:1015843517762
  38. TEERANACHAIDEEKUL V, MULLER R, JUNYAPRASERT V, Encapsulation of ascorbyl palmitate in nanostructured lipid carriers (NLC)—Effects of formulation parameters on physicochemical stability, 10.1016/j.ijpharm.2007.03.022
  39. Trevaskis Natalie L., Charman William N., Porter Christopher J.H., Lipid-based delivery systems and intestinal lymphatic drug transport: A mechanistic update, 10.1016/j.addr.2007.09.007
  40. Venishetty Vinay Kumar, Chede Raghavendra, Komuravelli Rojarani, Adepu Laxminarayana, Sistla Ramakrishna, Diwan Prakash V., Design and evaluation of polymer coated carvedilol loaded solid lipid nanoparticles to improve the oral bioavailability: A novel strategy to avoid intraduodenal administration, 10.1016/j.colsurfb.2012.01.001
  41. Williams Hywel D., Sassene Philip, Kleberg Karen, Bakala-N'Goma Jean-Claude, Calderone Marilyn, Jannin Vincent, Igonin Annabel, Partheil Anette, Marchaud Delphine, Jule Eduardo, Vertommen Jan, Maio Mario, Blundell Ross, Benameur Hassan, Carrière Frédéric, Müllertz Anette, Porter Christopher J.H., Pouton Colin W., Toward the Establishment of Standardized In Vitro Tests for Lipid-Based Formulations, Part 1: Method Parameterization and Comparison of In Vitro Digestion Profiles Across a Range of Representative Formulations, 10.1002/jps.23205
  42. Zhang Xiaoyong, Yin Jilei, Kang Cheng, Li Jing, Zhu Ying, Li Wenxin, Huang Qing, Zhu Zhiyong, Biodistribution and toxicity of nanodiamonds in mice after intratracheal instillation, 10.1016/j.toxlet.2010.07.001