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Displaying 15 results.
    • Journal article
    Mechanism-based thrombin inhibitors: design, synthesis, and molecular docking of a new selective 2-oxo-2H-1-benzopyran derivative.
    Frédérick, Raphaël[UCL] Robert, S.[FUNDP] Charlier, Caroline[FUNDP] Wouters, Johan[FUNDP] Masereel, Bernard[FUNDP] Pochet, Lionel[FUNDP] (2007) Journal of medicinal chemistry — Vol. 50, no. 15, p. 3645-3650 (2007)
    • Journal article
    Investigation of mechanism-based thrombin inhibitors: Implications of a highly conserved water molecule for the binding of coumarins within the S pocket.
    Frédérick, Raphaël[UCL] Charlier, Caroline[FUNDP] Robert, S.[FUNDP] Wouters, Johan[FUNDP] Masereel, Bernard[FUNDP] Pochet, Lionel[FUNDP] (2006) Bioorganic & Medicinal Chemistry Letters : the tetrahedron journal for research at the interface of chemistry and biology — Vol. 16, no. 7, p. 2017-2021 (2006)
    • Journal article
    3,6-disubstituted coumarins as mechanism-based inhibitors of thrombin and factor Xa
    Frédérick, Raphaël[UCL] Robert, S.[FUNDP] Charlier, Caroline[FUNDP] de Ruyck, Jérôme Wouters, Johan[FUNDP] Pirotte, Bernard Masereel, Bernard[FUNDP] Pochet, Lionel[FUNDP] (2005) Journal of Medicinal Chemistry — Vol. 48, no. 24, p. 7592-7603 (2005)
    • Journal article
    Chemical reactivity of plasma polymerized allylamine (PPAA) thin films on Au and Si : study of the thickness influence and aging of the films
    Moreau, Nicolas[FUNDP] Feron, Olivier[UCL] Gallez, Bernard[UCL] Masereel, Bernard[FUNDP] Michiels, Carine[FUNDP] Vander Borght, Thierry Rossi, François Lucas, Stéphane[FUNDP] (2011) Surface and Coatings Technology — Vol. 205, no. Suppl 2, p. S462-S465 (2011)
    • Journal article
    Antibody immobilization on gold nanoparticles coated layer-by-layer with polyelectrolytes
    Masereel, Bernard Dinguizli, Mustapha[FUNDP] Bouzin, Caroline[UCL] Moniotte, Nicolas[FUNDP] Feron, Olivier[UCL] Gallez, Bernard[UCL] Vander Borght, Thierry[UCL] Michiels , Carine[FUNDP] Lucas, Stéphane[FUNDP] (2011) Journal of Nanoparticle Research : an interdisciplinary forum for nanoscale science and technology — Vol. 13, no. 4, p. 1573-1580 (2011)
    • Journal article
    Tryptophan 2,3-dioxygenase (TDO) inhibitors. 3-(2-(pyridyl)ethenyl)indoles as potential anticancer immunomodulators
    Dolusic, Eduard[FUNDP] Larrieu, Pierre[UCL] Moineaux, Laurence[FUNDP] Stroobant, Vincent[UCL] Pilotte, Luc[UCL] Colau, Didier[UCL] Pochet, Lionel[FUNDP] Van den Eynde, Benoît[UCL] Masereel, Bernard[FUNDP] Wouters, Johan[FUNDP] Frédérick, Raphaël[FUNDP] (2011) Journal of Medicinal Chemistry — Vol. 54, no. 15, p. 5320-5334 (11/08/2011)
    • Journal article
    Design, solid-phase synthesis, and biological evaluation of novel 1,5-diarylpyrrole-3-carboxamides as carbonic anhydrase IX inhibitors
    Gluszok, Sebastien Frédérick, Raphaël[UCL] Foulon, Catherine Klupsch, Frederique Supuran, Claudiu T. Vullo, Daniela Scozzafava, Andrea Goossens, Jean-Francois Masereel, Bernard[FUNDP] Depreux, Patrick Goossens, Laurence (2010) Bioorganic & Medicinal Chemistry : the tetrahedron journal for research at the interface of chemistry and biology — Vol. 18, no. 21, p. 7392-7401 (2010)
    • Journal article
    Investigation of the inhibition mechanism of coumarins on chymotrypsin by mass spectrometry
    Pochet, Lionel[FUNDP] Dieu, Marc[FUNDP] Frédérick, Raphaël[UCL] Murray, Anne-Marie[FUNDP] Kempen, Isabelle Pirotte, Bernad Masereel, Bernard[FUNDP] (2003) Tetrahedron — Vol. 59, no. 25, p. 4557-4561 (2003)
    • Journal article
    Coumarin and isocoumarin as serine protease inhibitors
    Pochet, Lionel[FUNDP] Frédérick, Raphaël[UCL] Masereel, Bernard[FUNDP] (2004) Current pharmaceutical design — Vol. 10, no. 30, p. 3781-3796 (2004)
    • Journal article
    Modulators of the coagulation cascade: focus and recent advances in inhibitors of tissue factor, factor VIIa and their complex
    Frédérick, Raphaël[UCL] Pochet, Lionel[FUNDP] Charlier, Caroline[FUNDP] Masereel, Bernard[FUNDP] (2005) Current medicinal chemistry — Vol. 12, no. 4, p. 397-417 (2005)
    • Journal article
    Ligand-based and structure-based virtual screening to identify carbonic anhydrase IX inhibitors
    Thiry, Anne[FUNDP] Ledecq, Marie[FUNDP] Cecchi, Alessandro Frédérick, Raphaël[UCL] Dogné, Jean-Michel[FUNDP] Supuran, Caudiu T Wouters, Johan[FUNDP] Masereel, Bernard[FUNDP] (2009) Bioorganic & medicinal chemistry — Vol. 17, no. 2, p. 553-557 (2009)
    • Journal article
    Indol-2-yl ethanones as novel indoleamine 2,3-dioxygenase (IDO) inhibitors
    Dolusic, Eduard[FUNDP] Larrieu, Pierre[UCL] Blanc, Sébastien Sapunaric, Frédéric Norberg, Bernadette[FUNDP] Moineaux, Laurence[FUNDP] Colette, Delphine Stroobant, Vincent[UCL] Pilotte, Luc[UCL] Colau, Didier[UCL] Ferain, Thierry Fraser, Graeme Galleni, Moreno Frère, Jean-Marie Masereel, Bernard[FUNDP] Van den Eynde, Benoît[UCL] Wouters, Johan[FUNDP] Frédérick, Raphaël[UCL] (2011) Bioorganic & Medicinal Chemistry — Vol. 19, no. 4, p. 1550-1561 (2011)
    • Journal article
    Discovery and preliminary SARs of keto-indoles as novel indoleamine 2,3-dioxygenase (IDO) inhibitors
    Dolusic, Eduard[FUNDP] Larrieu, Pierre[UCL] Blanc, Sébastien Sapunaric, Frédéric Pouyez, Jenny[FUNDP] Moineaux, Laurence[FUNDP] Colette, Delphine Stroobant, Vincent[UCL] Pilotte, Luc[UCL] Colau, Didier[UCL] Ferain, Thierry Fraser, Graeme Galleni, Moreno Frère, Jean-Marie Masereel, Bernard[FUNDP] Van den Eynde, Benoît[UCL] Wouters, Johan[FUNDP] Frédérick, Raphaël[UCL] (2011) European Journal of Medicinal Chemistry — Vol. 46, no. 7, p. 3058-3065 (2011)
    • Journal article
    Corrigendum to "Indol-2-yl ethanones as novel indoleamine 2,3-dioxygenase (IDO) inhibitors" (Bioorganic and Medicinal Chemistry (2011) (1550-1561))
    Dolusic, Eduard[FUNDP] Larrieu, Pierre[UCL] Blanc, Sébastien Sapunaric, Frédéric Norberg, Bernadette[FUNDP] Moineaux, Laurence[FUNDP] Colette, Delphine Stroobant, Vincent[UCL] Pilotte, Luc[UCL] Colau, Didier[UCL] Ferain, Thierry Fraser, Graeme Galleni, Moreno Frre, Jean-Marie Masereel, Bernard[FUNDP] Van den Eynde, Benoît[UCL] Wouters, Johan[FUNDP] Frédérick, Raphaël[UCL] (2011) Bioorganic & Medicinal Chemistry : the tetrahedron journal for research at the interface of chemistry and biology — Vol. 19, no.9, p. 3029 (2011)
    • Journal article
    A comparison of six major platelet functional tests to assess the impact of carbon nanomaterials on platelet function: A practical guide.
    Mullier, François[UCL] Laloy, Julie Alpan, Lutfiye Mejia, Jorge Lucas, Stéphane Chatelain, Bernard Toussaint, Olivier Masereel, Bernard Rolin, Stéphanie Dogné, Jean-Michel (2013) Nanotoxicology — Vol. 8, no. 2, p. 220-232 (2013)