All Publications

Pages

1. • Journal article

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   The importance of screening solid-state phases of a racemic modification of a chiral drug: thermodynamic and structural characterization of solid-state phases of etiracetam

   Herman, Christelle Vermylen, Valérie Norberg, Bernadette[FUNDP] Wouters, Johan[FUNDP] Leyssens, Tom[UCL] (2013) Acta Crystallographica, Section B — Vol. B69, no. --, p. 371-378 (2013)
2. • Journal article

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   Structural study of prolinium/fumaric acid zwitterionic cocrystals: Focus on hydrogen-bonding pattern involving zwitterionic (Ionic) heterosynthons

   Tilborg, Anaëlle Leyssens, Tom[UCL] Norberg, Bernadette Wouters, Johan (2013) Crystal Growth and Design — Vol. 13, no.6, p. 2373-2389 (2013)
3. • Journal article

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   (3R, 5S, 6R, 8S, 9S)-1-Azonia-9-ethyl-3-hydroxy5-(6-methoxyquinolin-4-yl)-3-methyl-4-oxatricyclo[6.2.2.0]dodecane trifluoromethanesulfonate: insight into the sterochemistry of the cyclization

   Antequera-Garcia, Gema Norberg, Bernadette Marko, Istvan[UCL] Wouters, Johan (2006) Acta Crystallographica Section E-structure Reports Online — Vol. 62, p. O2864-O2865 (2006)
4. • Speech

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   Effective co-crystal screening through structural resemblance (poster)

   Springuel, Géraldine[UCL] Norberg, Bernadette[FUNDP] Robeyns, Koen[UCL] Wouters, Johan[FUNDP] Leyssens, Tom[UCL] (2011) International Symposium on Industrial Crystallization (ISIC18) — Zurich (Switzerland)
5. • Journal article

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   Structural insight into cocrystallization with zwitterionic co-formers: Cocrystals of S-naproxen

   Tumanova, Natalia[UCL] Tumanov, Nikolay[UCL] Robeyns, Koen[UCL] Filinchuk, Yaroslav[UCL] Wouters, Johan Leyssens, Tom[UCL] (2014) CrystEngComm — Vol. 16, no. 35, p. 8185-8196 (2014)
6. • Journal article

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   New bounds on right-handed currents from a polarization asymmetry correlation measurement with In-107

   Severijns, N. Gimeno-Nogues, F. Pepe, I. Wouters, Johan[FUNDP] Quin, P.A. Allet, M. Naviliat-Cuncic, O. De Moor, P. Schuurmans, P. Siebelink, R. Vanderpoorten, W. Vanhaverbeke, J. Vanneste, L. Prieels, René Deutsch, Jules (1992)
7. • Speech

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   Solid state chemistry of proline-Naproxen complexes (poster)

   Tilborg, Anaëlle[FUNDP] Springuel, Géraldine[UCL] Norberg, Bernadette[FUNDP] Leyssens, Tom[UCL] Wouters, Johan[FUNDP] (2012) 7th Belgian Crystallography Symposium (BCS-7) — Brussels (Belgium)
8. • Journal article

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   Versatile access to benzhydryl-phenylureas through an unexpected rearrangement during microwave-enhanced synthesis of hydantoins.

   Muccioli, Giulio[UCL] Wouters, Johan Poupaert, Jacques[UCL] Norberg, Bernadette Poppitz, Wolfgang Scriba, Gerhard K E Lambert, Didier[UCL] (2003) Organic letters — Vol. 5, no. 20, p. 3599-602 (2003)
9. • Journal article

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   Effects of Empirical Dispersion Energy on the Geometrical Parameters and Relative Energy of a Salicylideneaniline Molecular Switch in the Solid State

   QUERTINMONT, Jean Leyssens, Tom[UCL] Wouters, Johan Champagne, Benoit (2018) Crystals — Vol. 8, no.3, p. 125 (2018)
10. • Journal article

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    Acidochromic spiropyran–merocyanine stabilisation in the solid state

    Seiler, Vanessa Kristina[UCL] Callebaut, Kevin[UCL] Robeyns, Koen[UCL] Tumanov Nicolay Wouters, Johan Champagne, Benoit Leyssens, Tom[UCL] (2018) CrystEngCom — (2018)
11. • Journal article

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    A nano-sized container for specific encapsulation of isolated water molecules

    Lavendomme, Roy Marcélis, Lionel[UCL] Wouters, Johan Luhmer, Michel Jabin, Ivan (2016) Chemical Communications — Vol. 52, p. 14109-14112 (2016)
12. • Journal article

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    Opening Pandora’s Box: Chirality, Polymorphism, and Stoichiometric Diversity in Flurbiprofen/Proline Cocrystals

    Tumanova, Natalia[UCL] Tumanov, Nikolai Robeyns, Koen[UCL] Fischer, Franziska Fusaro, Luca Morelle, Fabrice[UCL] Ban, Voramsky Hautier, Geoffroy[UCL] Filinchuk, Yaroslav[UCL] Wouters, Johan Leyssens, Tom[UCL] Emmerling, Franziska (2018) Crystal Growth & Design — Vol. 18, no.2, p. 954-961 (2018)
13. • Journal article

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    A Structural Analysis of Spiropyran and Spirooxazine Compounds and Their Polymorphs

    Seiler, Vanessa Kristina[UCL] Tumanov, Nikolai Robeyns, Koen[UCL] Wouters, Johan Champagne, Benoit Leyssens, Tom[UCL] (2017) Crystals — Vol. 7, p. 84-95 (2017)
14. • Journal article

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    Direct Access by Mechanochemistry or Sonochemistry to Protonated Merocyanines: Components of a Four-State Molecular Switch

    Colaço, Melwin Carletta, Andrea Van Gysel, Mégane Robeyns, Koen[UCL] Tumanov, Nikolay Wouters, Johan (2018) ChemistryOpen — Vol. 7, no.7, p. 520-526 (2018)
15. • Journal article

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    Synthesis, evaluation and structure-activity relationship of new 3-carboxamide coumarins as FXIIa inhibitors

    Bouckaert, Charlotte[FUNDP] Serra, Silvia[FUNDP] Rondelet, Grégoire[FUNDP] Dolušić, Eduard[FUNDP] Wouters, Johan[FUNDP] Dogné, Jean-Michel[FUNDP] Frédérick, Raphaël[UCL] Pochet, Lionel[FUNDP] (2016) European Journal of Medicinal Chemistry — Vol. 110, p. 181-194 (2016)
16. • Journal article

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    A Study of Fasoracetam’s Solid State Forms: A Potential Anti-Alzheimer Pharmaceutical

    Harmsen, Bram[UCL] Robeyns, Koen[UCL] Wouters, Johan Leyssens, Tom[UCL] (2017) Journal of Pharmaceutical Sciences — Vol. 106, no.5, p. 1317-1321 (2017)
17. • Journal article

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    3D-QSAR, design, synthesis and characterization of trisubstituted harmine derivatives with in vitro antiproliferative properties

    Meinguet, Céline Bruyère, Céline Frédérick, Raphaël[UCL] Mathieu, Véronique Vancraeynest, Christelle Pochet, Lionel Laloy, Julie Mortier, Jérémie Wolber, Gerhard Kiss, Robert Masereel, Bernard Wouters, Johan (2015) European Journal of Medicinal Chemistry — Vol. 94, no. 1, p. 45-55 (2015)
18. • Journal article

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    Indol-2-yl ethanones as novel indoleamine 2,3-dioxygenase (IDO) inhibitors

    Dolusic, Eduard[FUNDP] Larrieu, Pierre[UCL] Blanc, Sébastien Sapunaric, Frédéric Norberg, Bernadette[FUNDP] Moineaux, Laurence[FUNDP] Colette, Delphine Stroobant, Vincent[UCL] Pilotte, Luc[UCL] Colau, Didier[UCL] Ferain, Thierry Fraser, Graeme Galleni, Moreno Frère, Jean-Marie Masereel, Bernard[FUNDP] Van den Eynde, Benoît[UCL] Wouters, Johan[FUNDP] Frédérick, Raphaël[UCL] (2011) Bioorganic & Medicinal Chemistry — Vol. 19, no. 4, p. 1550-1561 (2011)
19. • Journal article

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    Reversal of tumoral immune resistance by inhibition of tryptophan 2,3-dioxygenase.

    Pilotte, Luc Larrieu, Pierre Stroobant, Vincent Colau, Didier Dolusic, Eduard Frédérick, Raphaël De Plaen, Etienne Uyttenhove, Catherine Wouters, Johan Masereel, Bernard Van den Eynde, Benoît[UCL] (2012) Proceedings of the National Academy of Sciences of the United States of America — Vol. 109, no. 7, p. 2497-2502 (2012)
20. • Journal article

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    Synthesis and evaluation of β-carboline derivatives as potential monoamine oxidase inhibitors

    Reniers, Jérémy[FUNDP] Robert, S.[FUNDP] Frédérick, Raphaël[UCL] Masereel, Bernard[FUNDP] Vincent, S.[FUNDP] Wouters, Johan[FUNDP] (2011) European Journal of Medicinal Chemistry — Vol. 19, no. 1, p. 134-144 (2011)
21. • Journal article

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    Novel trisubstituted harmine derivatives with original in vitro anticancer activity

    Frédérick, Raphaël[UCL] Bruyére, Céline Vancraeynest, Christelle[FUNDP] Reniers, Jérémy[FUNDP] Meinguet, Céline[FUNDP] Pochet, Lionel[FUNDP] Backlund, Anders Masereel, Bernard[FUNDP] Kiss, Robert Wouters, Johan[FUNDP] (2012) Journal of Medicinal Chemistry — Vol. 55, no. 14, p. 6489-6501 (2012)
22. • Journal article

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    Thiosemicarbazide, a fragment with promising indolamine-2,3-dioxygenase (IDO) inhibition properties

    Serra, Silvia[FUNDP] Moineaux, Laurence[FUNDP] Vancraeynest, Christelle[FUNDP] Masereel, Bernard[FUNDP] Wouters, Johan[FUNDP] Pochet, Lionel[FUNDP] Frédérick, Raphaël[UCL] (2014) European Journal of Medicinal Chemistry — Vol. 82, p. 96-105 (2014)
23. • Journal article

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    Synthesis and inhibition study of monoamine oxidase, indoleamine 2,3-dioxygenase and tryptophan 2,3-dioxygenase by 3,8-substituted 5H-indeno[1,2-c]pyridazin-5-one derivatives

    Reniers, Jérémy[FUNDP] Meinguet, Céline[UCL] Moineaux, Laurence[FUNDP] Masereel, Bernard[FUNDP] Vincent, S.P. Frédérick, Raphaël[UCL] Wouters, Johan[FUNDP] (2011) European Journal of Medicinal Chemistry — Vol. 46, no. 12, p. 6104-6111 (2011)
24. • Journal article

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    Pyrazolo[4,3-c]isoquinolines as potential inhibitors of NF-κB activation

    Mortier, Jérémie[FUNDP] Frédérick, Raphaël[UCL] Ganeff, Corinne Remouchamps, Caroline Talaga, Patrice Pochet, Lionel[FUNDP] Wouters, Johan[FUNDP] Piette, Jacques Dejardin, Emmanuel Masereel, Bernard[FUNDP] (2010) Biochemical Pharmacology — Vol. 79, no. 10, p. 1462-1472 (2010)
25. • Journal article

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    Discovery and preliminary SARs of keto-indoles as novel indoleamine 2,3-dioxygenase (IDO) inhibitors

    Dolusic, Eduard[FUNDP] Larrieu, Pierre[UCL] Blanc, Sébastien Sapunaric, Frédéric Pouyez, Jenny[FUNDP] Moineaux, Laurence[FUNDP] Colette, Delphine Stroobant, Vincent[UCL] Pilotte, Luc[UCL] Colau, Didier[UCL] Ferain, Thierry Fraser, Graeme Galleni, Moreno Frère, Jean-Marie Masereel, Bernard[FUNDP] Van den Eynde, Benoît[UCL] Wouters, Johan[FUNDP] Frédérick, Raphaël[UCL] (2011) European Journal of Medicinal Chemistry — Vol. 46, no. 7, p. 3058-3065 (2011)

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