All Publications

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1. • Speech

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   A dual thromboxane inhibitor and thromboxane receptor antagonist prevents pig myocardial infarction induced by coronary thrombosis

   Rolin, S. Petein, M. Tchana-Sato, V. Dogne, Jean-Michel[UCL] Lambermont, B. Ghuysen, A. Kolh, P Masereel, Bernard[FUNDP] (2003) Congress of the European-Society-of-Cardiology — VIENNA(Austria)
2. • Journal article

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   Development of a PIXE analysis method for the determination of the biopersistence of SiC and TiC nanoparticles in rat lungs

   Lozano, Omar[FUNDP] Mejia, Jorge[FUNDP] Masereel, Bernard[FUNDP] Toussaint, Olivier[FUNDP] Lison, Dominique[UCL] Lucas, Stéphane[FUNDP] (2012) Nanotoxicology — Vol. 6, no. 3, p. 263-271 (2012)
3. • Journal article

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   3D-QSAR, design, synthesis and characterization of trisubstituted harmine derivatives with in vitro antiproliferative properties

   Meinguet, Céline Bruyère, Céline Frédérick, Raphaël[UCL] Mathieu, Véronique Vancraeynest, Christelle Pochet, Lionel Laloy, Julie Mortier, Jérémie Wolber, Gerhard Kiss, Robert Masereel, Bernard Wouters, Johan (2015) European Journal of Medicinal Chemistry — Vol. 94, no. 1, p. 45-55 (2015)
4. • Journal article

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   Indol-2-yl ethanones as novel indoleamine 2,3-dioxygenase (IDO) inhibitors

   Dolusic, Eduard[FUNDP] Larrieu, Pierre[UCL] Blanc, Sébastien Sapunaric, Frédéric Norberg, Bernadette[FUNDP] Moineaux, Laurence[FUNDP] Colette, Delphine Stroobant, Vincent[UCL] Pilotte, Luc[UCL] Colau, Didier[UCL] Ferain, Thierry Fraser, Graeme Galleni, Moreno Frère, Jean-Marie Masereel, Bernard[FUNDP] Van den Eynde, Benoît[UCL] Wouters, Johan[FUNDP] Frédérick, Raphaël[UCL] (2011) Bioorganic & Medicinal Chemistry — Vol. 19, no. 4, p. 1550-1561 (2011)
5. • Journal article

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   Reversal of tumoral immune resistance by inhibition of tryptophan 2,3-dioxygenase.

   Pilotte, Luc Larrieu, Pierre Stroobant, Vincent Colau, Didier Dolusic, Eduard Frédérick, Raphaël De Plaen, Etienne Uyttenhove, Catherine Wouters, Johan Masereel, Bernard Van den Eynde, Benoît[UCL] (2012) Proceedings of the National Academy of Sciences of the United States of America — Vol. 109, no. 7, p. 2497-2502 (2012)
6. • Journal article

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   Synthesis and evaluation of β-carboline derivatives as potential monoamine oxidase inhibitors

   Reniers, Jérémy[FUNDP] Robert, S.[FUNDP] Frédérick, Raphaël[UCL] Masereel, Bernard[FUNDP] Vincent, S.[FUNDP] Wouters, Johan[FUNDP] (2011) European Journal of Medicinal Chemistry — Vol. 19, no. 1, p. 134-144 (2011)
7. • Journal article

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   Novel trisubstituted harmine derivatives with original in vitro anticancer activity

   Frédérick, Raphaël[UCL] Bruyére, Céline Vancraeynest, Christelle[FUNDP] Reniers, Jérémy[FUNDP] Meinguet, Céline[FUNDP] Pochet, Lionel[FUNDP] Backlund, Anders Masereel, Bernard[FUNDP] Kiss, Robert Wouters, Johan[FUNDP] (2012) Journal of Medicinal Chemistry — Vol. 55, no. 14, p. 6489-6501 (2012)
8. • Journal article

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   Thiosemicarbazide, a fragment with promising indolamine-2,3-dioxygenase (IDO) inhibition properties

   Serra, Silvia[FUNDP] Moineaux, Laurence[FUNDP] Vancraeynest, Christelle[FUNDP] Masereel, Bernard[FUNDP] Wouters, Johan[FUNDP] Pochet, Lionel[FUNDP] Frédérick, Raphaël[UCL] (2014) European Journal of Medicinal Chemistry — Vol. 82, p. 96-105 (2014)
9. • Journal article

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   Synthesis and inhibition study of monoamine oxidase, indoleamine 2,3-dioxygenase and tryptophan 2,3-dioxygenase by 3,8-substituted 5H-indeno[1,2-c]pyridazin-5-one derivatives

   Reniers, Jérémy[FUNDP] Meinguet, Céline[UCL] Moineaux, Laurence[FUNDP] Masereel, Bernard[FUNDP] Vincent, S.P. Frédérick, Raphaël[UCL] Wouters, Johan[FUNDP] (2011) European Journal of Medicinal Chemistry — Vol. 46, no. 12, p. 6104-6111 (2011)
10. • Journal article

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    Pyrazolo[4,3-c]isoquinolines as potential inhibitors of NF-κB activation

    Mortier, Jérémie[FUNDP] Frédérick, Raphaël[UCL] Ganeff, Corinne Remouchamps, Caroline Talaga, Patrice Pochet, Lionel[FUNDP] Wouters, Johan[FUNDP] Piette, Jacques Dejardin, Emmanuel Masereel, Bernard[FUNDP] (2010) Biochemical Pharmacology — Vol. 79, no. 10, p. 1462-1472 (2010)
11. • Journal article

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    Discovery and preliminary SARs of keto-indoles as novel indoleamine 2,3-dioxygenase (IDO) inhibitors

    Dolusic, Eduard[FUNDP] Larrieu, Pierre[UCL] Blanc, Sébastien Sapunaric, Frédéric Pouyez, Jenny[FUNDP] Moineaux, Laurence[FUNDP] Colette, Delphine Stroobant, Vincent[UCL] Pilotte, Luc[UCL] Colau, Didier[UCL] Ferain, Thierry Fraser, Graeme Galleni, Moreno Frère, Jean-Marie Masereel, Bernard[FUNDP] Van den Eynde, Benoît[UCL] Wouters, Johan[FUNDP] Frédérick, Raphaël[UCL] (2011) European Journal of Medicinal Chemistry — Vol. 46, no. 7, p. 3058-3065 (2011)
12. • Journal article

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    Tryptophan 2,3-dioxygenase (TDO) inhibitors. 3-(2-(pyridyl)ethenyl)indoles as potential anticancer immunomodulators

    Dolusic, Eduard[FUNDP] Larrieu, Pierre[UCL] Moineaux, Laurence[FUNDP] Stroobant, Vincent[UCL] Pilotte, Luc[UCL] Colau, Didier[UCL] Pochet, Lionel[FUNDP] Van den Eynde, Benoît[UCL] Masereel, Bernard[FUNDP] Wouters, Johan[FUNDP] Frédérick, Raphaël[FUNDP] (2011) Journal of Medicinal Chemistry — Vol. 54, no. 15, p. 5320-5334 (11/08/2011)
13. • Journal article

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    New selective carbonic anhydrase IX inhibitors: Synthesis and pharmacological evaluation of diarylpyrazole-benzenesulfonamides

    Rogez-Florent, Tiphaine Meignan, Samuel Foulon, Catherine Six, Perrine Gros, Abigaëlle Bal-Mahieu, Christine Supuran, Claudiu T. Scozzafava, Andrea Frédérick, Raphaël[UCL] Masereel, Bernard[FUNDP] Depreux, Patrick Lansiaux, Amélie Goossens, Jean-François Gluszok, Sébastien Goossens, Laurence (2013) Bioorganic & Medicinal Chemistry : the tetrahedron journal for research at the interface of chemistry and biology — Vol. 21, no. 6, p. 1451-1464 (2013)
14. • Journal article

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    Indoleamine 2,3-dioxygenase inhibitory activity of derivatives of marine alkaloid tsitsikammamine A.

    Dolusic, Eduard[FUNDP] Larrieu, Pierre[UCL] Meinguet, Céline[FUNDP] Colette, Delphine Rives, Arnaud Blanc, Sébastien Ferain, Thierry Pilotte, Luc[UCL] Stroobant, Vincent[UCL] Wouters, Johan[FUNDP] Van den Eynde, Benoît[UCL] Masereel, Bernard[FUNDP] Delfourne, Evelyne Frédérick, Raphaël[UCL] (2013) Bioorganic & Medicinal Chemistry Letters — Vol. 23, no.1, p. 47-54 (2013)
15. • Journal article

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    Design, solid-phase synthesis, and biological evaluation of novel 1,5-diarylpyrrole-3-carboxamides as carbonic anhydrase IX inhibitors

    Gluszok, Sebastien Frédérick, Raphaël[UCL] Foulon, Catherine Klupsch, Frederique Supuran, Claudiu T. Vullo, Daniela Scozzafava, Andrea Goossens, Jean-Francois Masereel, Bernard[FUNDP] Depreux, Patrick Goossens, Laurence (2010) Bioorganic & Medicinal Chemistry : the tetrahedron journal for research at the interface of chemistry and biology — Vol. 18, no. 21, p. 7392-7401 (2010)
16. • Journal article

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    Corrigendum to "Indol-2-yl ethanones as novel indoleamine 2,3-dioxygenase (IDO) inhibitors" (Bioorganic and Medicinal Chemistry (2011) (1550-1561))

    Dolusic, Eduard[FUNDP] Larrieu, Pierre[UCL] Blanc, Sébastien Sapunaric, Frédéric Norberg, Bernadette[FUNDP] Moineaux, Laurence[FUNDP] Colette, Delphine Stroobant, Vincent[UCL] Pilotte, Luc[UCL] Colau, Didier[UCL] Ferain, Thierry Fraser, Graeme Galleni, Moreno Frre, Jean-Marie Masereel, Bernard[FUNDP] Van den Eynde, Benoît[UCL] Wouters, Johan[FUNDP] Frédérick, Raphaël[UCL] (2011) Bioorganic & Medicinal Chemistry : the tetrahedron journal for research at the interface of chemistry and biology — Vol. 19, no.9, p. 3029 (2011)
17. • Journal article

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    Synthesis, crystal structures and electronic properties of isomers of chloro-pyridinylvinyl-1H-indoles

    Moineaux, Laurence[FUNDP] Laurent, Sophie Reniers, Jérémy[FUNDP] Dolušić, Eduard[FUNDP] Galleni, Moreno Frère, Jean-Marie Masereel, Bernard[FUNDP] Frédérick, Raphaël[UCL] Wouters, Johan[FUNDP] (2012) European Journal of Medicinal Chemistry — Vol. 54, no. 1, p. 95-102 (2012)
18. • Journal article

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    NF-κB inducing kinase (NIK) inhibitors: Identification of new scaffolds using virtual screening

    Mortier, Jérémie[FUNDP] Masereel, Bernard[FUNDP] Remouchamps, Caroline Ganeff, Corinne Piette, Jacques Frédérick, Raphaël[UCL] (2010) Bioorganic & Medicinal Chemistry Letters : the tetrahedron journal for research at the interface of chemistry and biology — Vol. 20, no. 15, p. 4515-4520 (2010)
19. • Journal article

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    Modulators of the coagulation cascade: focus and recent advances in inhibitors of tissue factor, factor VIIa and their complex

    Frédérick, Raphaël[UCL] Pochet, Lionel[FUNDP] Charlier, Caroline[FUNDP] Masereel, Bernard[FUNDP] (2005) Current medicinal chemistry — Vol. 12, no. 4, p. 397-417 (2005)
20. • Journal article

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    Coumarin and isocoumarin as serine protease inhibitors

    Pochet, Lionel[FUNDP] Frédérick, Raphaël[UCL] Masereel, Bernard[FUNDP] (2004) Current pharmaceutical design — Vol. 10, no. 30, p. 3781-3796 (2004)
21. • Journal article

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    Ligand-based and structure-based virtual screening to identify carbonic anhydrase IX inhibitors

    Thiry, Anne[FUNDP] Ledecq, Marie[FUNDP] Cecchi, Alessandro Frédérick, Raphaël[UCL] Dogné, Jean-Michel[FUNDP] Supuran, Caudiu T Wouters, Johan[FUNDP] Masereel, Bernard[FUNDP] (2009) Bioorganic & medicinal chemistry — Vol. 17, no. 2, p. 553-557 (2009)
22. • Journal article

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    Investigation of the inhibition mechanism of coumarins on chymotrypsin by mass spectrometry

    Pochet, Lionel[FUNDP] Dieu, Marc[FUNDP] Frédérick, Raphaël[UCL] Murray, Anne-Marie[FUNDP] Kempen, Isabelle Pirotte, Bernad Masereel, Bernard[FUNDP] (2003) Tetrahedron — Vol. 59, no. 25, p. 4557-4561 (2003)
23. • Journal article

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    Synthesis and anticonvulsant activity of 2(3H)-benzoxazolone and 2(3H)-benzothiazolone derivatives.

    Ucar, H Van derpoorten, K Cacciaguerra, S Spampinato, S Stables, J P Depovere, Paul[UCL] Isa, M. Masereel, Bernard[FUNDP] Delarge, J. Poupaert, Jacques[UCL] (1998) Journal of medicinal chemistry — Vol. 41, no. 7, p. 1138-45 (1998)
24. • Journal article

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    Synthesis and biological evaluation of a new family of anti-benzylanilinosulfonamides as CA IX inhibitors.

    Thiry, Anne Delayen, Aurélie Goossens, Laurence Houssin, Raymond Ledecq, Marie Frankart, A. Dogné, Jean-Michel Wouters, Johan Supuran, Claudiu T Hénichart, Jean-Pierre Masereel, Bernard[FUNDP] (2008) European journal of medicinal chemistry — Vol. 44, no. 2, p. 511-8 (2009)
25. • Journal article

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    "Fries like" rearrangement: a novel and efficient method for the synthesis of 6-acyl-2(3H)-benzoxazolones and 6-acyl-2(3H)-benzothiazolones

    Ucar, H Van Derpoorten, K Depovere, Paul[UCL] Lesieur, D. Isa, M. Masereel, Bernard[FUNDP] Delarge, J. Poupaert, Jacques[UCL] (1998) Tetrahedron — Vol. 54, no. 9, p. 1763-1772 (1998)

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