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1. • Article de périodique

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   A MBP-FAAH fusion protein as a tool to produce human and rat fatty acid amide hydrolase : expression and pharmacological comparison

   Labar, Geoffray[UCL] Vliet, Françoise V. Wouters, Johan[FUNDP] Lambert, Didier[UCL] (2008) Amino Acids — Vol. 34, no. 1, p. 127-133 (2008)
2. • Article de périodique

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   Short, asymmetric synthesis of epi-morphine ACNO analogues.

   Heureux, Nicolas[UCL] Wouters, Johan Norberg, Bernadette Marko, Istvan[UCL] (2006) Organic & biomolecular chemistry — Vol. 4, no. 21, p. 3898-900 (2006)
3. • Article de périodique

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   Disulfiram is an inhibitor of human purified monoacylglycerol lipase, the enzyme regulating 2-arachidonoylglycerol signaling

   Labar, Geoffray[UCL] Bauvois, Cedric[UCL] Muccioli, Giulio[UCL] Wouters, Johan[FUNDP] Lambert, Didier[UCL] (2007) ChemBioChem — Vol. 8, no. 11, p. 1293-1297 (2007)
4. • Article de périodique

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   Sequential acid/base-catalyzed polycyclization of tryptamine derivatives. A rapid access to Büchi's ketone.

   Heureux, Nicolas[UCL] Wouters, Johan Marko, Istvan[UCL] (2005) Organic letters — Vol. 7, no. 23, p. 5245-8 (2005)
5. • Article de périodique

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   1-Benzhydryl-3-phenylurea and 1-benzhydryl-3-phenylthiourea derivatives: new templates among the CB1 cannabinoid receptor inverse agonists.

   Muccioli, Giulio[UCL] Wouters, Johan Scriba, Gerhard K E Poppitz, Wolfgang Poupaert, Jacques[UCL] Lambert, Didier[UCL] (2005) Journal of medicinal chemistry — Vol. 48, no. 23, p. 7486-90 (2005)
6. • Article de périodique

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   Engineering Solid-State Molecular Switches: N-Salicylidene N-Heterocycle Derivatives

   Robert, François[UCL] Naik, Anil[UCL] Hidara, Florence[UCL] Tinant, Bernard[UCL] Robiette, Raphaël[UCL] Wouters, Johan Garcia, Yann[UCL] (2010) European Journal of Organic Chemistry — , no. 4, p. 621-637 (2010)
7. • Article de périodique

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   A Review on the Monoacylglycerol Lipase : at the Interface between Fat and Endocannabinoid Signalling

   Labar, Geoffray[UCL] Wouters, Johan[FUNDP] Lambert, Didier[UCL] (2010) Current Medicinal Chemistry — Vol. 17, no. 24, p. 2588-2607 (2010)
8. • Article de périodique

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   Copper-Catalysed Domino Silylative Aldol Reaction Leading to Stereocontrolled Chiral Quaternary Carbons.

   Welle, Alexandre[UCL] Petrignet, Julien Tinant, Bernard[UCL] Wouters, Johan Riant, Olivier[UCL] (2010) Chemistry (Weinheim an der Bergstrasse, Germany) — Vol. 16, no. 36, p. 10980-3 (2010)
9. • Article de périodique

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   Crystal Structure of the Human Monoacylglycerol Lipase, a Key Actor in Endocannabinoid Signaling.

   Labar, Geoffray[UCL] Bauvois, Cédric Borel, Franck Ferrer, Jean-Luc Wouters, Johan[FUNDP] Lambert, Didier[UCL] (2010) ChemBioChem — Vol. 11, no. 2, p. 218-227 (2010)
10. • Article de périodique

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    Mechanism-based thrombin inhibitors: design, synthesis, and molecular docking of a new selective 2-oxo-2H-1-benzopyran derivative.

    Frédérick, Raphaël[UCL] Robert, S.[FUNDP] Charlier, Caroline[FUNDP] Wouters, Johan[FUNDP] Masereel, Bernard[FUNDP] Pochet, Lionel[FUNDP] (2007) Journal of medicinal chemistry — Vol. 50, no. 15, p. 3645-3650 (2007)
11. • Article de périodique

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    Investigation of mechanism-based thrombin inhibitors: Implications of a highly conserved water molecule for the binding of coumarins within the S pocket.

    Frédérick, Raphaël[UCL] Charlier, Caroline[FUNDP] Robert, S.[FUNDP] Wouters, Johan[FUNDP] Masereel, Bernard[FUNDP] Pochet, Lionel[FUNDP] (2006) Bioorganic & Medicinal Chemistry Letters : the tetrahedron journal for research at the interface of chemistry and biology — Vol. 16, no. 7, p. 2017-2021 (2006)
12. • Article de périodique

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    3,6-disubstituted coumarins as mechanism-based inhibitors of thrombin and factor Xa

    Frédérick, Raphaël[UCL] Robert, S.[FUNDP] Charlier, Caroline[FUNDP] de Ruyck, Jérôme Wouters, Johan[FUNDP] Pirotte, Bernard Masereel, Bernard[FUNDP] Pochet, Lionel[FUNDP] (2005) Journal of Medicinal Chemistry — Vol. 48, no. 24, p. 7592-7603 (2005)
13. • Article de périodique

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    Convenient one-pot formation of highly functionalized 5-bromo-2-aminothiazoles, potential endocannabinoid hydrolase MAGL inhibitors

    Prevost, Julien R.C.[UCL] Kozlova, Arina[UCL] Es Saadi, Bouazza[UCL] Yildiz, Esra[UCL] Modaffari, Sara Lambert, Didier M.[UCL] Pochet, Lionel Wouters, Johan Dolušić, Eduard Frédérick, Raphaël[UCL] (2018) Tetrahedron Letters — Vol. 59, no.49, p. 4315-4319 (2018)
14. • Article de périodique

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    Improving Nefiracetam Dissolution and Solubility Behavior Using a Cocrystallization Approach

    Buol, Xavier[UCL] Robeyns, Koen[UCL] Caro Garrido, Camila[UCL] TUMANOV, Nikolay Collard, Laurent[UCL] Wouters, Johan Leyssens, Tom[UCL] (2020) Pharmaceutics — Vol. 12, no.7, p. 653 (2020)
15. • Article de périodique

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    Pharmacomodulations of the benzoyl-thiosemicarbazide scaffold reveal antimicrobial agents targeting D-alanyl-D-alanine ligase in bacterio

    Ameryckx, Alice[UCL] Pochet, Lionel Wang, Gang[UCL] Yildiz, Esra[UCL] Es Saadi, Bouazza[UCL] Wouters, Johan Van Bambeke, Françoise[UCL] Frédérick, Raphaël[UCL] (2020) European Journal of Medicinal Chemistry — Vol. 200, no.1, p. 112444 (2020)
16. • Article de périodique

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    1-(2-Hydroxybenzoyl)-thiosemicarbazides are promising antimicrobial agents targeting d-alanine-d-alanine ligase in bacterio

    Ameryckx, Alice[UCL] Thabault, Léopold[UCL] Pochet, Lionel Leimanis, Serge Poupaert, Jacques[UCL] Wouters, Johan Joris, Bernard Van Bambeke, Françoise[UCL] Frédérick, Raphaël[UCL] (2018) European Journal of Medicinal Chemistry — Vol. 159, p. 324-338 (2018)
17. • Article de périodique

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    Chiral Resolution of Mandelic Acid through Preferential Cocrystallization with Nefiracetam

    Buol, Xavier[UCL] Caro Garrido, Camila[UCL] Robeyns, Koen[UCL] Tumanov, Nikolay Collard, Laurent[UCL] Wouters, Johan Leyssens, Tom[UCL] (2020) Crystal Growth & Design — Vol. 20, no.12, p. 7979-7988 (2020)
18. • Article de périodique

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    Transmembrane (TMEM) protein family members: Poorly characterized even if essential for the metastatic process.

    Marx, Sébastien Dal Maso, Thomas Chen, Jia-Wei Bury, Marina[UCL] Wouters, Johan Michiels, Carine Le Calvé, Benjamin (2020) Seminars in cancer biology — Vol. 60, p. 96-106 (2020)
19. • Article de périodique

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    Combining API in a dual-drug ternary cocrystal approach

    Song, Lixing[UCL] Robeyns, Koen[UCL] Tumanov, Nikolay Wouters, Johan Leyssens, Tom[UCL] (2020) Chemical Communications — Vol. 56, no.86, p. 13229-13232 (2020)
20. • Article de périodique

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    Sterically hindered ortho-substituted phosphatriptycenes as configurationally stable P-chirogenic triarylphosphines

    Hu, Lei[UCL] Mahaut, Damien Tumanov, Nikolay Wouters, Johan Collard, Laurent[UCL] Robiette, Raphaël[UCL] Berionni, Guillaume (2021) Dalton Transactions — Vol. 50, no.14, p. 4772-4777 (2021)
21. • Article de périodique

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    Unraveling the Effects of Co-Crystallization on the UV/Vis Absorption Spectra of an N-Salicylideneaniline Derivative. A Computational RI-CC2 Investigation

    QUERTINMONT, Jean Leyssens, Tom[UCL] Wouters, Johan Champagne, Benoit (2020) Molecules — Vol. 25, no.19, p. 4512 (2020)
22. • Article de périodique

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    Combining Two Antitubercular Drugs, Clofazimine and 4-Aminosalicylic Acid, in Order to Improve Clofazimine Aqueous Solubility and 4-Aminosalicylic Acid Thermal Stability

    BODART, Laurie DERLET, Amélie Buol, Xavier[UCL] Leyssens, Tom[UCL] TUMANOV, Nikolay Wouters, Johan (2020) Journal of Pharmaceutical Sciences — Vol. 109, no.12, p. 3645-3652 (2020)
23. • Article de périodique

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    Synthesis and anticonvulsant activity of N,N-phthaloyl derivatives of central nervous system inhibitory amino acids

    Usifoh, CO Lambert, DM. Wouters, Johan[FUNDP] Scriba, GKE. (2001) Archiv der Pharmazie — Vol. 334, no. 10, p. 323-331 (2001)
24. • Article de périodique

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    A rapid and efficient microwave-assisted synthesis of hydantoins and thiohydantoins

    Muccioli, Giulio[UCL] Poupaert, Jacques[UCL] Wouters, Johan Norberg, Bernadette Poppitz, Wolfgang Scriba, Gerhard K. E. Lambert, Didier[UCL] (2003) Tetrahedron — Vol. 59, no. 8, p. 1301-1307 (2003)
25. • Article de périodique

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    In-beam Induced Nuclear-polarization of Radioactive Ion-beams

    Wouters, Johan[FUNDP] Vanderpoorten, W. Silverans, R. Schuurmans, P. Demoor, P. Vanneste, L. Vervier, Jean[UCL] (1991) Nuclear Instruments & Methods in Physics Research. Section B: Beam Interactions with Materials and Atoms — Vol. 61, no. 3, p. 348-356 (1991)

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