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1. • Brevet

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   [18F]-labelled lactate derivative as PET radiotracer

   Sonveaux, Pierre[UCL] Labar, Daniel[UCL] Van Hee, Vincent F[UCL] Dehon, Gwenaël[UCL] Frédérick, Raphaël[UCL] (2018)
2. • Article de périodique

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   Synthesis, evaluation and structure-activity relationship of new 3-carboxamide coumarins as FXIIa inhibitors

   Bouckaert, Charlotte[FUNDP] Serra, Silvia[FUNDP] Rondelet, Grégoire[FUNDP] Dolušić, Eduard[FUNDP] Wouters, Johan[FUNDP] Dogné, Jean-Michel[FUNDP] Frédérick, Raphaël[UCL] Pochet, Lionel[FUNDP] (2016) European Journal of Medicinal Chemistry — Vol. 110, p. 181-194 (2016)
3. • Article de périodique

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   Synthesis and in vitro evaluation of polyethylene glycol paclitaxel conjugates for lung cancer therapy

   Luo, Tian[UCL] Magnusson, J Préat, Véronique[UCL] Frédérick, Raphaël[UCL] Alexander, Cameron Bosquillon, Cynthia Vanbever, Rita[UCL] (2016) Pharmaceutical Research — Vol. 33, no. 7, p. 1671-1681
4. • Article de périodique

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   Computational tools for in silico fragment-based drug design

   Mortier, Jeremie Rakers, Christin Frédérick, Raphaël[UCL] Wolber, Gerhard (2012) Current Topics in Medicinal Chemistry — Vol. 12, no. 17, p. 1935-1943 (2012)
5. • Article de périodique

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   Synthesis and biological evaluation of di-aryl urea derivatives as c-Kit inhibitors

   Ravez, Séverine Arsenlis, Stéphane Barczyk, Amélie Dupont, Anthony Frédérick, Raphaël[UCL] Hesse, Stéphanie Kirsch, Gilbert Depreux, Patrick Goossens, Laurence (2015) Bioorganic & Medicinal Chemistry : the tetrahedron journal for research at the interface of chemistry and biology — Vol. 23, no.22, p. 7340-7347 (2015)
6. • Article de périodique

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   Novel pyrazolo[1,5-a]pyridines as PI3K inhibitors: variation of the central linker group

   Kendall, Jackie D. Marshall, Andrew J. Giddens, Anna C. Tsang, Kit Yee Boyd, Maruta Frédérick, Raphaël[UCL] Lill, Claire L. Lee, Woo-Jeong Kolekar, Sharada Chao, Mindy Malik, Alisha Yu, Shuqiao Chaussade, Claire Buchanan, Christina M. Rewcastle, Gordon W. Baguley, Bruce C. Flanagan, Jack U. Denny, William A. Shepherd, Peter R. (2014) MedChemComm — Vol. 5, no.1, p. 41 [1-6] (2014)
7. • Article de périodique

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   Indoleamine 2,3-dioxygenase inhibitors: a patent review (2008 - 2012).

   Dolusic, Eduard Frédérick, Raphaël[UCL] (2013) Expert Opinion on Therapeutic Patents — Vol. 23, no.10, p. 1367-1381 (2013)
8. • Article de périodique

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   3D-QSAR, design, synthesis and characterization of trisubstituted harmine derivatives with in vitro antiproliferative properties

   Meinguet, Céline Bruyère, Céline Frédérick, Raphaël[UCL] Mathieu, Véronique Vancraeynest, Christelle Pochet, Lionel Laloy, Julie Mortier, Jérémie Wolber, Gerhard Kiss, Robert Masereel, Bernard Wouters, Johan (2015) European Journal of Medicinal Chemistry — Vol. 94, no. 1, p. 45-55 (2015)
9. • Article de périodique

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   Indol-2-yl ethanones as novel indoleamine 2,3-dioxygenase (IDO) inhibitors

   Dolusic, Eduard[FUNDP] Larrieu, Pierre[UCL] Blanc, Sébastien Sapunaric, Frédéric Norberg, Bernadette[FUNDP] Moineaux, Laurence[FUNDP] Colette, Delphine Stroobant, Vincent[UCL] Pilotte, Luc[UCL] Colau, Didier[UCL] Ferain, Thierry Fraser, Graeme Galleni, Moreno Frère, Jean-Marie Masereel, Bernard[FUNDP] Van den Eynde, Benoît[UCL] Wouters, Johan[FUNDP] Frédérick, Raphaël[UCL] (2011) Bioorganic & Medicinal Chemistry — Vol. 19, no. 4, p. 1550-1561 (2011)
10. • Article de périodique

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    Reversal of tumoral immune resistance by inhibition of tryptophan 2,3-dioxygenase.

    Pilotte, Luc Larrieu, Pierre Stroobant, Vincent Colau, Didier Dolusic, Eduard Frédérick, Raphaël De Plaen, Etienne Uyttenhove, Catherine Wouters, Johan Masereel, Bernard Van den Eynde, Benoît[UCL] (2012) Proceedings of the National Academy of Sciences of the United States of America — Vol. 109, no. 7, p. 2497-2502 (2012)
11. • Article de périodique

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    Synthesis and evaluation of β-carboline derivatives as potential monoamine oxidase inhibitors

    Reniers, Jérémy[FUNDP] Robert, S.[FUNDP] Frédérick, Raphaël[UCL] Masereel, Bernard[FUNDP] Vincent, S.[FUNDP] Wouters, Johan[FUNDP] (2011) European Journal of Medicinal Chemistry — Vol. 19, no. 1, p. 134-144 (2011)
12. • Article de périodique

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    Novel trisubstituted harmine derivatives with original in vitro anticancer activity

    Frédérick, Raphaël[UCL] Bruyére, Céline Vancraeynest, Christelle[FUNDP] Reniers, Jérémy[FUNDP] Meinguet, Céline[FUNDP] Pochet, Lionel[FUNDP] Backlund, Anders Masereel, Bernard[FUNDP] Kiss, Robert Wouters, Johan[FUNDP] (2012) Journal of Medicinal Chemistry — Vol. 55, no. 14, p. 6489-6501 (2012)
13. • Article de périodique

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    Thiosemicarbazide, a fragment with promising indolamine-2,3-dioxygenase (IDO) inhibition properties

    Serra, Silvia[FUNDP] Moineaux, Laurence[FUNDP] Vancraeynest, Christelle[FUNDP] Masereel, Bernard[FUNDP] Wouters, Johan[FUNDP] Pochet, Lionel[FUNDP] Frédérick, Raphaël[UCL] (2014) European Journal of Medicinal Chemistry — Vol. 82, p. 96-105 (2014)
14. • Article de périodique

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    Synthesis and inhibition study of monoamine oxidase, indoleamine 2,3-dioxygenase and tryptophan 2,3-dioxygenase by 3,8-substituted 5H-indeno[1,2-c]pyridazin-5-one derivatives

    Reniers, Jérémy[FUNDP] Meinguet, Céline[UCL] Moineaux, Laurence[FUNDP] Masereel, Bernard[FUNDP] Vincent, S.P. Frédérick, Raphaël[UCL] Wouters, Johan[FUNDP] (2011) European Journal of Medicinal Chemistry — Vol. 46, no. 12, p. 6104-6111 (2011)
15. • Article de périodique

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    Pyrazolo[4,3-c]isoquinolines as potential inhibitors of NF-κB activation

    Mortier, Jérémie[FUNDP] Frédérick, Raphaël[UCL] Ganeff, Corinne Remouchamps, Caroline Talaga, Patrice Pochet, Lionel[FUNDP] Wouters, Johan[FUNDP] Piette, Jacques Dejardin, Emmanuel Masereel, Bernard[FUNDP] (2010) Biochemical Pharmacology — Vol. 79, no. 10, p. 1462-1472 (2010)
16. • Article de périodique

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    Discovery and preliminary SARs of keto-indoles as novel indoleamine 2,3-dioxygenase (IDO) inhibitors

    Dolusic, Eduard[FUNDP] Larrieu, Pierre[UCL] Blanc, Sébastien Sapunaric, Frédéric Pouyez, Jenny[FUNDP] Moineaux, Laurence[FUNDP] Colette, Delphine Stroobant, Vincent[UCL] Pilotte, Luc[UCL] Colau, Didier[UCL] Ferain, Thierry Fraser, Graeme Galleni, Moreno Frère, Jean-Marie Masereel, Bernard[FUNDP] Van den Eynde, Benoît[UCL] Wouters, Johan[FUNDP] Frédérick, Raphaël[UCL] (2011) European Journal of Medicinal Chemistry — Vol. 46, no. 7, p. 3058-3065 (2011)
17. • Article de périodique

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    Radiosynthesis and validation of (±)-[18F]-3-fluoro-2-hydroxypropionate ([18F]-FLac) as a PET tracer of lactate to monitor MCT1-dependent lactate uptake in tumors

    Van Hee, Vincent F[UCL] Labar, Daniel[UCL] Dehon, Gwenaël[UCL] Grasso, Debora[UCL] Gregoire, Vincent[UCL] Muccioli, Giulio[UCL] Frédérick, Raphaël[UCL] Sonveaux, Pierre[UCL] (2017) OncoTarget — Vol. 8, no. 15, p. 24415-24428 (2017)
18. • Article de périodique

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    Insight into the Diels-Alder reaction : A green chemistry revisitation of the synthesis of a cantharidine-like trypanocidal pilot-molecule

    Gbaguidi, Fernand A. Kassehin, Comlan Urbain[UCL] Prévost, Julien[UCL] Frédérick, Raphaël[UCL] McCurdy, Christopher R. Poupaert, Jacques[UCL] (2015) Journal of Chemical and Pharmaceutical Research — Vol. 7, no.7, p. 1109-1113 (2015)
19. • Article de périodique

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    Tryptophan 2,3-dioxygenase (TDO) inhibitors. 3-(2-(pyridyl)ethenyl)indoles as potential anticancer immunomodulators

    Dolusic, Eduard[FUNDP] Larrieu, Pierre[UCL] Moineaux, Laurence[FUNDP] Stroobant, Vincent[UCL] Pilotte, Luc[UCL] Colau, Didier[UCL] Pochet, Lionel[FUNDP] Van den Eynde, Benoît[UCL] Masereel, Bernard[FUNDP] Wouters, Johan[FUNDP] Frédérick, Raphaël[FUNDP] (2011) Journal of Medicinal Chemistry — Vol. 54, no. 15, p. 5320-5334 (11/08/2011)
20. • Article de périodique

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    Synthesis and biological evaluation of novel analogues of the pan class i phosphatidylinositol 3-kinase (PI3K) inhibitor 2-(Difluoromethyl)-1-[4,6-di(4- morpholinyl)-1,3,5-triazin-2-yl]-1 H -benzimidazole (ZSTK474)

    Rewcastle, Gordon W. Gamage, Swarna A. Flanagan, Jack U. Frédérick, Raphaël[UCL] Denny, William A. Baguley, Bruce C. Kestell, Philip Singh, Ripudaman Kendall, Jackie D. Marshall, Elaine S. Lill, Claire L. Lee, Woo-Jeong Kolekar, Sharada Buchanan, Christina M. Jamieson, Stephen M.F. Shepherd, Peter R. (2011) Journal of Medicinal Chemistry — Vol. 54, no.20, p. 7105-7126 (2011)
21. • Article de périodique

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    New selective carbonic anhydrase IX inhibitors: Synthesis and pharmacological evaluation of diarylpyrazole-benzenesulfonamides

    Rogez-Florent, Tiphaine Meignan, Samuel Foulon, Catherine Six, Perrine Gros, Abigaëlle Bal-Mahieu, Christine Supuran, Claudiu T. Scozzafava, Andrea Frédérick, Raphaël[UCL] Masereel, Bernard[FUNDP] Depreux, Patrick Lansiaux, Amélie Goossens, Jean-François Gluszok, Sébastien Goossens, Laurence (2013) Bioorganic & Medicinal Chemistry : the tetrahedron journal for research at the interface of chemistry and biology — Vol. 21, no. 6, p. 1451-1464 (2013)
22. • Article de périodique

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    Indoleamine 2,3-dioxygenase inhibitory activity of derivatives of marine alkaloid tsitsikammamine A.

    Dolusic, Eduard[FUNDP] Larrieu, Pierre[UCL] Meinguet, Céline[FUNDP] Colette, Delphine Rives, Arnaud Blanc, Sébastien Ferain, Thierry Pilotte, Luc[UCL] Stroobant, Vincent[UCL] Wouters, Johan[FUNDP] Van den Eynde, Benoît[UCL] Masereel, Bernard[FUNDP] Delfourne, Evelyne Frédérick, Raphaël[UCL] (2013) Bioorganic & Medicinal Chemistry Letters — Vol. 23, no.1, p. 47-54 (2013)
23. • Article de périodique

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    Design, solid-phase synthesis, and biological evaluation of novel 1,5-diarylpyrrole-3-carboxamides as carbonic anhydrase IX inhibitors

    Gluszok, Sebastien Frédérick, Raphaël[UCL] Foulon, Catherine Klupsch, Frederique Supuran, Claudiu T. Vullo, Daniela Scozzafava, Andrea Goossens, Jean-Francois Masereel, Bernard[FUNDP] Depreux, Patrick Goossens, Laurence (2010) Bioorganic & Medicinal Chemistry : the tetrahedron journal for research at the interface of chemistry and biology — Vol. 18, no. 21, p. 7392-7401 (2010)
24. • Article de périodique

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    Corrigendum to "Indol-2-yl ethanones as novel indoleamine 2,3-dioxygenase (IDO) inhibitors" (Bioorganic and Medicinal Chemistry (2011) (1550-1561))

    Dolusic, Eduard[FUNDP] Larrieu, Pierre[UCL] Blanc, Sébastien Sapunaric, Frédéric Norberg, Bernadette[FUNDP] Moineaux, Laurence[FUNDP] Colette, Delphine Stroobant, Vincent[UCL] Pilotte, Luc[UCL] Colau, Didier[UCL] Ferain, Thierry Fraser, Graeme Galleni, Moreno Frre, Jean-Marie Masereel, Bernard[FUNDP] Van den Eynde, Benoît[UCL] Wouters, Johan[FUNDP] Frédérick, Raphaël[UCL] (2011) Bioorganic & Medicinal Chemistry : the tetrahedron journal for research at the interface of chemistry and biology — Vol. 19, no.9, p. 3029 (2011)
25. • Article de périodique

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    Synthesis, crystal structures and electronic properties of isomers of chloro-pyridinylvinyl-1H-indoles

    Moineaux, Laurence[FUNDP] Laurent, Sophie Reniers, Jérémy[FUNDP] Dolušić, Eduard[FUNDP] Galleni, Moreno Frère, Jean-Marie Masereel, Bernard[FUNDP] Frédérick, Raphaël[UCL] Wouters, Johan[FUNDP] (2012) European Journal of Medicinal Chemistry — Vol. 54, no. 1, p. 95-102 (2012)

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