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Affichage: 5 résultats.
    • Article de périodique
    Discovery of pyrazolo[1,5-a]pyridines as p110α-selective PI3 kinase inhibitors
    Kendall, Jackie D. O'Connor, Patrick D. Marshall, Andrew J. Frédérick, Raphaël[UCL] Marshall, Elaine S. Lill, Claire L. Lee, Woo-Jeong Kolekar, Sharada Chao, Mindy Malik, Alisha Yu, Shuqiao Chaussade, Claire Buchanan, Christina Rewcastle, Gordon W. Baguley, Bruce C. Flanagan, Jack U. Jamieson, Stephen M.F. Denny, William A. Shepherd, Peter R. (2012) Bioorganic & Medicinal Chemistry : the tetrahedron journal for research at the interface of chemistry and biology — Vol. 20, no. 1, p. 69-85 (2012)
    • Article de périodique
    Synthesis and biological evaluation of novel analogues of the pan class i phosphatidylinositol 3-kinase (PI3K) inhibitor 2-(Difluoromethyl)-1-[4,6-di(4- morpholinyl)-1,3,5-triazin-2-yl]-1 H -benzimidazole (ZSTK474)
    Rewcastle, Gordon W. Gamage, Swarna A. Flanagan, Jack U. Frédérick, Raphaël[UCL] Denny, William A. Baguley, Bruce C. Kestell, Philip Singh, Ripudaman Kendall, Jackie D. Marshall, Elaine S. Lill, Claire L. Lee, Woo-Jeong Kolekar, Sharada Buchanan, Christina M. Jamieson, Stephen M.F. Shepherd, Peter R. (2011) Journal of Medicinal Chemistry — Vol. 54, no.20, p. 7105-7126 (2011)
    • Article de périodique
    Novel pyrazolo[1,5-a]pyridines as p110α-selective PI3 kinase inhibitors: Exploring the benzenesulfonohydrazide SAR
    Kendall, Jackie D. Giddens, Anna C. Tsang, Kit Yee Frédérick, Raphaël[UCL] Marshall, Elaine S. Singh, Ripudaman Lill, Claire L. Lee, Woo-Jeong Kolekar, Sharada Chao, Mindy Malik, Alisha Yu, Shuqiao Chaussade, Claire Buchanan, Christina Rewcastle, Gordon W. Baguley, Bruce C. Flanagan, Jack U. Jamieson, Stephen M.F. Denny, William A. Shepherd, Peter R. (2012) Bioorganic & Medicinal Chemistry : the tetrahedron journal for research at the interface of chemistry and biology — Vol. 20, no. 1, p. 58-68 (2012)
    • Article de périodique
    Phosphoinositide-3-kinases (PI3Ks): Combined comparative modeling and 3D-QSAR to rationalize the inhibition of p110α
    Frédérick, Raphaël[UCL] Denny, William A. (2008) Journal of Chemical Information and Modeling — Vol. 48, no. 3, p. 629-638 (2008)
    • Article de périodique
    Novel pyrazolo[1,5-a]pyridines as PI3K inhibitors: variation of the central linker group
    Kendall, Jackie D. Marshall, Andrew J. Giddens, Anna C. Tsang, Kit Yee Boyd, Maruta Frédérick, Raphaël[UCL] Lill, Claire L. Lee, Woo-Jeong Kolekar, Sharada Chao, Mindy Malik, Alisha Yu, Shuqiao Chaussade, Claire Buchanan, Christina M. Rewcastle, Gordon W. Baguley, Bruce C. Flanagan, Jack U. Denny, William A. Shepherd, Peter R. (2014) MedChemComm — Vol. 5, no.1, p. 41 [1-6] (2014)