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1. • Journal article

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   Mechanism-based thrombin inhibitors: design, synthesis, and molecular docking of a new selective 2-oxo-2H-1-benzopyran derivative.

   Frédérick, Raphaël[UCL] Robert, S.[FUNDP] Charlier, Caroline[FUNDP] Wouters, Johan[FUNDP] Masereel, Bernard[FUNDP] Pochet, Lionel[FUNDP] (2007) Journal of medicinal chemistry — Vol. 50, no. 15, p. 3645-3650 (2007)
2. • Journal article

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   Investigation of mechanism-based thrombin inhibitors: Implications of a highly conserved water molecule for the binding of coumarins within the S pocket.

   Frédérick, Raphaël[UCL] Charlier, Caroline[FUNDP] Robert, S.[FUNDP] Wouters, Johan[FUNDP] Masereel, Bernard[FUNDP] Pochet, Lionel[FUNDP] (2006) Bioorganic & Medicinal Chemistry Letters : the tetrahedron journal for research at the interface of chemistry and biology — Vol. 16, no. 7, p. 2017-2021 (2006)
3. • Journal article

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   3,6-disubstituted coumarins as mechanism-based inhibitors of thrombin and factor Xa

   Frédérick, Raphaël[UCL] Robert, S.[FUNDP] Charlier, Caroline[FUNDP] de Ruyck, Jérôme Wouters, Johan[FUNDP] Pirotte, Bernard Masereel, Bernard[FUNDP] Pochet, Lionel[FUNDP] (2005) Journal of Medicinal Chemistry — Vol. 48, no. 24, p. 7592-7603 (2005)
4. • Journal article

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   Bioavailability and anticonvulsant activity of 2-cyanoguanidinophenytoin, a structural analogue of phenytoin

   Lambert, Didier[UCL] Masereel, Bernard Gallez, Bernard[UCL] Geurts, Muriel[UCL] Scriba, Gerhard K. E. (1996) Journal of Pharmaceutical Sciences — Vol. 85, no. 10, p. 1077-1081 (1996)
5. • Journal article

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   Evidence for a neuroprotective effect of pyrid-3-yl-sulphonyl-urea in photochemically induced focal ischaemia in rats: magnetic resonance imaging evaluation.

   Baudelet, Christine[UCL] Demeure, R. Frois, A Masereel, Bernard[FUNDP] Goudemant, Jean-François[UCL] Ritter, Christian[UCL] Gallez, Bernard[UCL] (1999) The Journal of pharmacy and pharmacology — Vol. 51, no. 8, p. 967-70 (1999)
6. • Speech

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   A dual thromboxane inhibitor and thromboxane receptor antagonist prevents pig myocardial infarction induced by coronary thrombosis

   Rolin, S. Petein, M. Tchana-Sato, V. Dogne, Jean-Michel[UCL] Lambermont, B. Ghuysen, A. Kolh, P Masereel, Bernard[FUNDP] (2003) Congress of the European-Society-of-Cardiology — VIENNA(Austria)
7. • Journal article

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   Anticonvulsant activity and interactions with neuronal voltage-dependent sodium channel of analogues of ameltolide

   Vamecq, J. Lambert, Didier[UCL] Poupaert, Jacques[UCL] Masereel, Bernard[FUNDP] Stables, JP. (1998) Journal of Medicinal Chemistry — Vol. 41, no. 18, p. 3307-13 (1998)
8. • Journal article

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   Validation of the calibrated thrombin generation test (cTGT) as the reference assay to evaluate the procoagulant activity of nanomaterials

   Laloy, Julie[FUNDP] Robert, S.[FUNDP] Marbehant, Catherine[FUNDP] Mullier, François[UCL] Mejia, Jorge[FUNDP] Piret, Jean-Pascal[FUNDP] Lucas, Stéphane[FUNDP] Chatelain, Bernard[UCL] Dogné, Jean-Michel[FUNDP] Toussaint, Olivier[FUNDP] Masereel, Bernard[FUNDP] Rolin, Stéphanie[FUNDP] (2012) Nanotoxicology — Vol. 6, no. 2, p. 213-232 (2012)
9. • Journal article

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   Development of a PIXE analysis method for the determination of the biopersistence of SiC and TiC nanoparticles in rat lungs

   Lozano, Omar[FUNDP] Mejia, Jorge[FUNDP] Masereel, Bernard[FUNDP] Toussaint, Olivier[FUNDP] Lison, Dominique[UCL] Lucas, Stéphane[FUNDP] (2012) Nanotoxicology — Vol. 6, no. 3, p. 263-271 (2012)
10. • Journal article

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    Tryptophan 2,3-dioxygenase (TDO) inhibitors. 3-(2-(pyridyl)ethenyl)indoles as potential anticancer immunomodulators

    Dolusic, Eduard[FUNDP] Larrieu, Pierre[UCL] Moineaux, Laurence[FUNDP] Stroobant, Vincent[UCL] Pilotte, Luc[UCL] Colau, Didier[UCL] Pochet, Lionel[FUNDP] Van den Eynde, Benoît[UCL] Masereel, Bernard[FUNDP] Wouters, Johan[FUNDP] Frédérick, Raphaël[FUNDP] (2011) Journal of Medicinal Chemistry — Vol. 54, no. 15, p. 5320-5334 (11/08/2011)
11. • Journal article

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    Synthesis, crystal structures and electronic properties of isomers of chloro-pyridinylvinyl-1H-indoles

    Moineaux, Laurence[FUNDP] Laurent, Sophie Reniers, Jérémy[FUNDP] Dolušić, Eduard[FUNDP] Galleni, Moreno Frère, Jean-Marie Masereel, Bernard[FUNDP] Frédérick, Raphaël[UCL] Wouters, Johan[FUNDP] (2012) European Journal of Medicinal Chemistry — Vol. 54, no. 1, p. 95-102 (2012)
12. • Journal article

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    Indoleamine 2,3-dioxygenase inhibitory activity of derivatives of marine alkaloid tsitsikammamine A.

    Dolusic, Eduard[FUNDP] Larrieu, Pierre[UCL] Meinguet, Céline[FUNDP] Colette, Delphine Rives, Arnaud Blanc, Sébastien Ferain, Thierry Pilotte, Luc[UCL] Stroobant, Vincent[UCL] Wouters, Johan[FUNDP] Van den Eynde, Benoît[UCL] Masereel, Bernard[FUNDP] Delfourne, Evelyne Frédérick, Raphaël[UCL] (2013) Bioorganic & Medicinal Chemistry Letters — Vol. 23, no.1, p. 47-54 (2013)
13. • Journal article

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    Design, solid-phase synthesis, and biological evaluation of novel 1,5-diarylpyrrole-3-carboxamides as carbonic anhydrase IX inhibitors

    Gluszok, Sebastien Frédérick, Raphaël[UCL] Foulon, Catherine Klupsch, Frederique Supuran, Claudiu T. Vullo, Daniela Scozzafava, Andrea Goossens, Jean-Francois Masereel, Bernard[FUNDP] Depreux, Patrick Goossens, Laurence (2010) Bioorganic & Medicinal Chemistry : the tetrahedron journal for research at the interface of chemistry and biology — Vol. 18, no. 21, p. 7392-7401 (2010)
14. • Journal article

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    New selective carbonic anhydrase IX inhibitors: Synthesis and pharmacological evaluation of diarylpyrazole-benzenesulfonamides

    Rogez-Florent, Tiphaine Meignan, Samuel Foulon, Catherine Six, Perrine Gros, Abigaëlle Bal-Mahieu, Christine Supuran, Claudiu T. Scozzafava, Andrea Frédérick, Raphaël[UCL] Masereel, Bernard[FUNDP] Depreux, Patrick Lansiaux, Amélie Goossens, Jean-François Gluszok, Sébastien Goossens, Laurence (2013) Bioorganic & Medicinal Chemistry : the tetrahedron journal for research at the interface of chemistry and biology — Vol. 21, no. 6, p. 1451-1464 (2013)
15. • Journal article

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    NF-κB inducing kinase (NIK) inhibitors: Identification of new scaffolds using virtual screening

    Mortier, Jérémie[FUNDP] Masereel, Bernard[FUNDP] Remouchamps, Caroline Ganeff, Corinne Piette, Jacques Frédérick, Raphaël[UCL] (2010) Bioorganic & Medicinal Chemistry Letters : the tetrahedron journal for research at the interface of chemistry and biology — Vol. 20, no. 15, p. 4515-4520 (2010)
16. • Journal article

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    Investigation of the inhibition mechanism of coumarins on chymotrypsin by mass spectrometry

    Pochet, Lionel[FUNDP] Dieu, Marc[FUNDP] Frédérick, Raphaël[UCL] Murray, Anne-Marie[FUNDP] Kempen, Isabelle Pirotte, Bernad Masereel, Bernard[FUNDP] (2003) Tetrahedron — Vol. 59, no. 25, p. 4557-4561 (2003)
17. • Journal article

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    Coumarin and isocoumarin as serine protease inhibitors

    Pochet, Lionel[FUNDP] Frédérick, Raphaël[UCL] Masereel, Bernard[FUNDP] (2004) Current pharmaceutical design — Vol. 10, no. 30, p. 3781-3796 (2004)
18. • Journal article

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    Modulators of the coagulation cascade: focus and recent advances in inhibitors of tissue factor, factor VIIa and their complex

    Frédérick, Raphaël[UCL] Pochet, Lionel[FUNDP] Charlier, Caroline[FUNDP] Masereel, Bernard[FUNDP] (2005) Current medicinal chemistry — Vol. 12, no. 4, p. 397-417 (2005)
19. • Journal article

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    Synthesis and biological evaluation of a new family of anti-benzylanilinosulfonamides as CA IX inhibitors.

    Thiry, Anne Delayen, Aurélie Goossens, Laurence Houssin, Raymond Ledecq, Marie Frankart, A. Dogné, Jean-Michel Wouters, Johan Supuran, Claudiu T Hénichart, Jean-Pierre Masereel, Bernard[FUNDP] (2008) European journal of medicinal chemistry — Vol. 44, no. 2, p. 511-8 (2009)
20. • Journal article

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    Synthesis and anticonvulsant activity of 2(3H)-benzoxazolone and 2(3H)-benzothiazolone derivatives.

    Ucar, H Van derpoorten, K Cacciaguerra, S Spampinato, S Stables, J P Depovere, Paul[UCL] Isa, M. Masereel, Bernard[FUNDP] Delarge, J. Poupaert, Jacques[UCL] (1998) Journal of medicinal chemistry — Vol. 41, no. 7, p. 1138-45 (1998)
21. • Journal article

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    "Fries like" rearrangement: a novel and efficient method for the synthesis of 6-acyl-2(3H)-benzoxazolones and 6-acyl-2(3H)-benzothiazolones

    Ucar, H Van Derpoorten, K Depovere, Paul[UCL] Lesieur, D. Isa, M. Masereel, Bernard[FUNDP] Delarge, J. Poupaert, Jacques[UCL] (1998) Tetrahedron — Vol. 54, no. 9, p. 1763-1772 (1998)
22. • Journal article

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    Ligand-based and structure-based virtual screening to identify carbonic anhydrase IX inhibitors

    Thiry, Anne[FUNDP] Ledecq, Marie[FUNDP] Cecchi, Alessandro Frédérick, Raphaël[UCL] Dogné, Jean-Michel[FUNDP] Supuran, Caudiu T Wouters, Johan[FUNDP] Masereel, Bernard[FUNDP] (2009) Bioorganic & medicinal chemistry — Vol. 17, no. 2, p. 553-557 (2009)
23. • Journal article

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    Indol-2-yl ethanones as novel indoleamine 2,3-dioxygenase (IDO) inhibitors

    Dolusic, Eduard[FUNDP] Larrieu, Pierre[UCL] Blanc, Sébastien Sapunaric, Frédéric Norberg, Bernadette[FUNDP] Moineaux, Laurence[FUNDP] Colette, Delphine Stroobant, Vincent[UCL] Pilotte, Luc[UCL] Colau, Didier[UCL] Ferain, Thierry Fraser, Graeme Galleni, Moreno Frère, Jean-Marie Masereel, Bernard[FUNDP] Van den Eynde, Benoît[UCL] Wouters, Johan[FUNDP] Frédérick, Raphaël[UCL] (2011) Bioorganic & Medicinal Chemistry — Vol. 19, no. 4, p. 1550-1561 (2011)
24. • Journal article

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    Synthesis and inhibition study of monoamine oxidase, indoleamine 2,3-dioxygenase and tryptophan 2,3-dioxygenase by 3,8-substituted 5H-indeno[1,2-c]pyridazin-5-one derivatives

    Reniers, Jérémy[FUNDP] Meinguet, Céline[UCL] Moineaux, Laurence[FUNDP] Masereel, Bernard[FUNDP] Vincent, S.P. Frédérick, Raphaël[UCL] Wouters, Johan[FUNDP] (2011) European Journal of Medicinal Chemistry — Vol. 46, no. 12, p. 6104-6111 (2011)
25. • Journal article

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    Thiosemicarbazide, a fragment with promising indolamine-2,3-dioxygenase (IDO) inhibition properties

    Serra, Silvia[FUNDP] Moineaux, Laurence[FUNDP] Vancraeynest, Christelle[FUNDP] Masereel, Bernard[FUNDP] Wouters, Johan[FUNDP] Pochet, Lionel[FUNDP] Frédérick, Raphaël[UCL] (2014) European Journal of Medicinal Chemistry — Vol. 82, p. 96-105 (2014)

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